Konferencje

1. Society of Applied Neuroscience & National Initiative Brain & Cognition, 30.01-02.02.2014, Utrecht, the Netherlands;

Chilmonczyk Z., Walory J., Bojarski A., Sylte I., Nowak G., Szewczyk B. Zinc and depresion. Modulation of serotonergic neurotransmission by zinc at a cellular level. BoA p81-82 Abstract

2. Barcelona GPCR Spring Conference 2014, 28-30.04.2014, Barcelona, Spain;

Warszycki, D.; Rueda, M.; Kristiansen, K.; Sylte, I.; Abagyan, R.; Bojarski, A.J. Ligand binding mode analysis using new 5-HT1A receptor models developed by ALiBERO methodology BoA p23 Poster
Mordalski, S.; Bojarski, A.J. 2D-SIFt – a matrix describing detailed interactions between ligand and receptor. BoA p31-32 Poster
Smusz, S.; Czarnecki, W.; Warszycki, D.; Bojarski, A.J. Uncertainty of the in vitro experiments in the predictive models construction. BoA p32-33 Poster
Rataj, K.; Czarnecki, W.; Smusz, S.; Bojarski, A.J. 2D fingerprints – a new way of chemical structure description. BoA p31 Poster

3. The Ninth Multidisciplinary Conference on Drug Research, 12-14.05.2014, Szydłów, Poland;

Chilmonczyk, Z; Sylte, I. Bojarski, A.J. Ligand-directed receptor trafficking. BoA p7 Abstract

4. The Ninth Multidisciplinary Conference on Drug Research, 12-14.05.2014, Szydłów, Poland;

Walory, J.; Sylte, I.; Bojarski, A.J.; Nowak, G; Chilmończyk, Z. Serotonin transporter inhibitors inducing hypotermia at mice. BoA p70 Abstract

5. GPCR Structure, Function and Drug Discovery Conference, 19-26.05.2014, Cambridge, USA;

Freyd, T.; Warszycki, D.; Gabrielsen, M.; Mordalski, S.; Kristiansen, K.; Chilmonczyk, Z.; Bojarski, A.J.; Sylte, I. Allosteric modulation of the human GABA B receptor. Abstract

6. The 5th Annual BioStruct Conference, 28–31.08.2014, Jægtvolden, Norway;

Freyd, T.; Warszycki, D.; Gabrielsen, M.; Kristiansen, K.; Chilmonczyk, Z.; Bojarski, A.J.; Sylte, I. Allosteric modulation of the human GABAB receptor: Development of a tool for antidepressant drug discovery. BoA p22 Abstract

7. The XXIII International Symposium on Medicinal Chemistry (EFMC-ISMC 2014), 07-11.09.2014, Lisbon, Portugal;

Jarończyk, M.; Chilmonczyk, Z.; Mazurek, A.P.; Bojarski, A.J.; Sylte, I. Binding of arylopiperazine derivatives to 5-HT1A serotonin receptor with new flexible docking approach. poster D 021
Walory, J.; Chilmonczyk, Z.; Bojarski, A.J.; Sylte, I.; Kossakowski, J.; Jarończyk, M. The influence of substituents on the ligand binding affinity to serotonin transporter. poster Y 069

8. VIth Conversatory on Medicinal Chemistry, 18-20.09.2014, Lublin, Poland;

Mordalski, S.; Bojarski, A.J. 2D-SIFt – a matrix describing ligand-receptor interactions. BoA p121 Abstract Poster
Warszycki, D.; Staroń, J.; Kafel, R.; Bojarski, A.J. Lessons learned from analysis of bioisosteric substitution in ligands of serotonin receptor family. BoA p188 Abstract Poster

9. The Schrödinger 14th Annual European User Meeting, 29.09-01.10.2014, Frankfurt, Germany;

Fidom, K.; Isberg, V.; Mordalski, S.; Hauser, A.; Lehto, T.; ; Bojarski, A.J.; Gloriam, D.E. A new crystal strycture fragment-based pharmacophore method for G Protein-Coupled receptors. BoA p84 Abstract

10. The GLISTEN Budapest 2014 Conference, 02-04.10.2014, Budapest, Hungary;

Mordalski, S.; Bojarski, A.J. Computational study on GPCR – G protein interfaces. BoA p15 Abstract
Rataj, K.; Witek. J.; Mordalski, S.; Bojarski, A.J. SIFt-guided agonist/antagonist differentiation for beta2-AR ligands. BoA p55 Abstract Poster
Warszycki, D.; Mordalski, S.; Freyd, T.; Sylte, I.; Bojarski, A.J. Pharmacophore modeling of GABA-B receptor ligands – methodology and application for virtual screening. BoA p53 Abstract Poster

11. Contacting meeting for the Norwegian Biochemical Society (NBS), 09-12.02.2015, Svaldbard, Norway;

Gabrielsen, M.; Kurczab, R.; Siwek, A.; Wolak, M.; Ravna, A.W.; Kristiansen, K.; Kufaraeva, I.; Abagyan, R.; Nowak, G.; Chilmonczyk, Z.; Sylte, I.; Bojarski, A.J.; Identification of Novel Serotonin Transporter Compounds by Virtual Screening and Experimental Verification. Book of Abstracts.
Freyd, T.; Warszycki, D.; Gabrielsen, M.; Mordalski, S.; Kristiansen, K.; Chilmonczyk, Z.; Bojarski, A.J.; Sylte, I.; Allosteric modulation of the human GABAB receptor. Book of Abstracts.

12. Annual meeting of the Norwegian Society of Pharmacology and Toxicology, 28-31.01.2015, Beito, Norway;

Gabrielsen, M.; Kurczab, R.; Siwek, A.; Wolak, M.; Ravna, A.W.; Kristiansen, K.; Kufaraeva, I.; Abagyan, R.; Nowak, G.; Chilmonczyk, Z.; Sylte, I.; Bojarski, A.J.; Identification of Novel Serotonin Transporter Compounds by Virtual Screening and Experimental Verification. Book of Abstracts.

13. GLISTEN Meeting 2015, 01-02.04.2015, Allschwil, Switzerland;

Hogendorf, A.; Satała, G.; Staroń, J.; Hogendorf, A.; Bugno, R.; Warszycki, D.; Bojarski, A.J.; Three point pharmacophore investigation leads to novel serotonergic chemotypes. BoA p44 Poster
Kurczab, R.; Canale, V. ; Zajdel, P.; Bojarski, A.J.; A step toward GPCRs polypharmacology: an algorithm to 5-HT7/5-HT1A selectivity prediction; BoA p56 Poster

14. Dokonania Naukowe Doktorantów III Edycja,.18.04.2015, Kraków, Poland;

Hogendorf, A.; Bugno, R.; Satała, G.; Hogendorf, A.; Staroń, J.; Warszycki, D.; Bojarski, A.J.; Design and synthesis of aminergic GPCR’s ligands. BoA p24 Abstract Poster
Hogendorf, A.; Bojarski, A.J.; Synthesis of indole derivatives as building blocks in organic and medicinal chemistry. BoA p23 Abstract Poster

15. BIT’s 8th Annual World Protein & Peptide Conference, 25-28.04.2015, Nanjing, China;

Chilmonczyk, Z.; Bojarski, A.J.; Sylte, I.; Functional selectivity and antidepressant activity of serotonin 1A receptor ligands; BoA Abstract

16. IXth Joint Meeting in Medicinal Chemistry, Athens, Greece, 2015.06.07-10;

Walory, J.; Koronkiewicz, M.; Bojarski, A.J.; Sylte, I.; Kossakowski, J.; Jarończyk, M.; Chilmonczyk, Z.; New SERT inhibitors with antineoplastic activity. Book of Abstracts.
Jarończyk, M.; Bojarski, A.J.; Sylte, I.; Chilmonczyk, Z.; The search for new ligands with dual activity for SERT and serotonin receptors. Book of Abstracts.

17. V Meeting of the Paul Ehrlich MedChem Euro-PhD Network, 03-05.07.2015, Kraków, Poland;

Hogendorf, A.; Brański, P.; Burnat, G.; Bugno, R.; Hogendorf, A.; Chruścicka, B.; Bojarski, A.J.; Finding Allosteric Modulators of Metabotropic Glutamate Receptors as Potential CNS Drugs. BoA P-15 Abstract Poster

18. VIIth Conversatory on Medicinal Chemistry, 17-19.09.2015, Lublin, Poland;

Wushur, I; Freyd, T. Evenseth, L.; Sylte, I.; Allosteric modulation of GABAB receptor. BoA K05 Abstract
Freyd, T.; Warszycki, D.; Gabrielsen, M.; Mordalski, S.; Kristiansen, K.; Chilmonczyk, Z.; Bojarski, A.J.; Sylte, I.; Allosteric modulation of the human GABAB receptor. BoA K08 Abstract
Chilmonczyk, Z.; Bojarski, A.; Sylte, I.; Participation of pre- and postsynaptic of 5-HT1A receptors in mood regulation (modulation of depressive like behaviours). BoA K 16 Abstract
Hogendorf, A.; Hogendorf, A.; Bojarski, A.J.; The synthesis of fused heterocyclic building blocks and their application as core structures of GPCR ligands. BoA P42 Abstract
Mordalski, S.; Bojarski, A.J.; An active conformation of mGlu2 receptor induced by molecular dynamics simulation with C-terminal Gi peptide. BoA P68 Abstract
Staroń, J.; Warszycki, D.; Satała, G.; Bojarski, A.J.; Derivatives of N-[2-(dimethylamine)ethyl]-N-(2-phenylethyl)-aniline as potential polypharmacological ligands of SERT/5-HT6/5-HT7. BoA P92 Abstract
Podlewska, S.; Kurczab, R.; Satała, G.; Bojarski, A.J.; New non-basic ligands of serotonin receptor 5-HT6 as a result of virtual screening based on machine-learning methods. BoA PP5 Abstract
Hogendorf, A.; Brański, P.; Burnat, G.; Bugno, R.; Hogendorf, A.; Chruścicka, B.; Bojarski, A.J.; The development of mGluR8 PAM agonists. BoA PP13 Abstract

19. 15th European Schrodinger User Group Meeting, 23-25.09.2015, Paris, France;

Mordalski, S.; Podolak, I.; Bojarski, A.J.; 2D-SIFt – a matrix describing detailed interactions between ligand and receptor. BOA p86 Poster

20. GLISTEN Meeting Amsterdam 2015, 12-13.10.2015, Amsterdam, The Netherlands;

Warszycki, D.; Kafel, R.; Bojarski, A.J.; Application of linear combination of pharmacophore hypotheses into search for the dual 5-T1A/SERT ligands. BoA p36 Abstract Poster
Rataj, K.; Czarnecki, W.; Podlewska, S.; Bojarski, A.J.; Structural Connectivity Fingerprints – a New Way to Represent and Classify Compounds. BoA p35 Abstract Poster
Mordalski, S.; Witek, J.; Podlewska, S.; Rataj, K.; Bojarski, A.J.; Multiple conformational states in retrospective virtual screening – homology models vs. crystal structures. ß2 adrenergic receptor case study. BoA p9 Abstract Poster
Podlewska, S.; Warszycki, D.; Bojarski, A.J.; Because two is always better than one – towards the search of dual 5-HTx-SERT ligands. BoA p25 Abstract Poster

21. 11th German Conference on Chemoinformatics, 08-10.11.2015, Fulda, Germany;

Kurczab, R.; Bojarski, A.J.; New approach for evaluation of docking results based on hybrid interaction fingerprint and machine learning methods. Book of Abstracts, p.P30.

22. GLISTEN Meeting 2016, 06-08.04.2016, Erlangen, Germany;

Mordalski, S.; Pocha, A.; Podolak, I.; Bojarski, A.J.; Application of SVM and 2D-SIFt into interaction-guided virtual screening. Book of Abstracts, P60

23. 10th Interdisciplinary Conference on Drug Research 15-18.05.2016, Korytnica, Poland;

Milczarek, M.; Wiktorska, K.; Śliwka, L.; Lubelska, K.; Matosiuk, D.; Chilmonczyk, Z.; Mechanism of synergic interaction between sulforaphane and 5-fluorouracil in the breast cell line MDA-MB- 231. Book of Abstracts,
Lubelska, K.; Wiktorska, K.; Śliwka, L.; Milczarek, M.; Chilmonczyk, Z.; Sulforaphane regulates differently NRF2 dependent induction of detoxification enzymes in normal and cancer colorectal cells. Book of Abstracts,
Wiktorska, K.; Śliwka, L.; Lubelska, K.; Milczarek, M.; Krug, P.; Cierpiał, T.; Kiełbasiński, P.; Suchocki, P.; Mazur, M.; Chilmonczyk, Z.; Sulforaphane analogs – new perspectives in cancer treatment? Book of Abstracts,
Śliwka, L.; Wiktorska, K.; Koronkiewicz, M.; Milczarek, M.; Lubelska, K.; Suchocki, P.; Chilmonczyk, Z.; The mechanism of synergism between selol and sulforaphane in the breast cancer cell line MCF-7. Book of Abstracts,

24. 2nd Central European Biomedical Congress (CEBC), 15-18.06.2016, Kraków, Poland;

Staroń, J.; Kurczab, R.; Warszycki, D.; Satała, G.; Bugno, R.; Hogendorf, A.; Bojarski, A.J.; Halogen bonding enhances affinity at 5-HT7R in a series of N-[2- (dimethylamine)ethyl]-N-(2-phenylehtyl)anilines. Book of Abstracts, p.135.

25. Polish Scientific Networks: Science and Business, 06.30-07.02.2016, Wrocław, Poland;

Staroń, J.; Warszycki, D.; Kurczab, R.; Satała, G.; Kalinowska-Tłuścik, J.; Bojarski, A.J.; Unexpected discoveries in the development of 5-HT6 receptor ligands. Book of Abstracts,

26. XXIV EFMC International Symposium on Medicinal Chemistry, 28.08-01.09.2016, Manchester, United Kingdom;

Hogendorf, A.S.; Hogendorf, A.; Kurczab, R.; Satała, G.; Lenda, T.; Latacz, G.; Bugno, R.; Staroń, J.; Bojarski, A.J.; Low-basicity 5-HT 7 agonists as potential molecular probes, PET-radiotracers or pharmacological drugs. Book of Abstracts,

27. 3rd EFMC Young Medicinal Chemist Symposium, 01-02.09.2016, Manchester, United Kingdom, Book of Abstracts;

Hogendorf, A.S.; Hogendorf, A.; Kurczab, R.; Satała, G.; Lenda, T.; Latacz, G.; Bugno, R.; Staroń, J.; Bojarski, A.J.; Determining the binding mode of 3-(1- alkyl-1H-imidazole- 5-yl)-1Hi-indole. Book of Abstracts,

28. VIIIth Conversatory on Medicinal Chemistry, 15-17.09.2016, Lublin, Poland;

Wushur, I.; Freyd, T.; Evenseth, L.M.; Gabrielsen, M.; Warszycki, D.; Mordalski, S.; Brański, P.; Chruścicka, B.; Burnat, G.; Pilc, A.; Bojarski, A.J.; Screening for GABAB receptor compounds. Book of Abstracts, NS1.
Hogendorf, A.S.; Hogendorf, A.; Kurczab, R.; Satała, G.; Lenda, T.; Latacz, G.; Bugno, R.; Staroń, J.; Bojarski, A.J.; Low-basicity agonists of 5-HT7 receptor synthesized by van Leusen multicomponent reaction. Book of Abstracts, NS2.
Walory, J.; Śliwka, L.; Chilmonczyk, Z.; Neuroprotective and proapoptotic activity of serotonin transporter inhibitors and serotonin receptor ligands. Book of Abstracts, NS3.
Kurczab, R.; Kafel, R.; Bojarski, A.J.; Development of a new methods for virtual screening protocol. Book of Abstracts, NS4.
Hogendorf, A.; Hogendorf, A.S.; Kurczab, R.; Satała, G.; Bojarski, A.J.; Binding mode analysis of a series of novel 5-HT1A ligands. Book of Abstracts, P4.
Evenseth, L.M.; Sylte,I.; Screening for novel GABAB orthosteric ligands, Book of Abstracts, P117
Freyd, T.; Warszycki, D.; Gabrielsen, M.; Mordalski, S.; Bojarski, A.J.; Sylte, I.; Allosteric modulation of the human GABAB receptor. Book of Abstracts, P118.

29. Glisten 2016 Prague, 26-17.09.2016, Prague, Czech Republic;

Freyd, T.; Evenseth, L.M.; Wushur, I.; Gabrielsen, M.; Warszycki, D.; Mordalski, S.; Brański, P.; Chruścicka, B.; Burnat, G.; Pilc, A.; Bojarski, A.J.; Sylte, I.; Screening for new GABAB receptor compounds.